Jacob J Plattner: search on Z-Library

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1

Topical treatment for cutaneous leishmaniasis – dermato-pharmacokinetic led optimisation of benzoxaboroles

Van Bocxlaer, Katrien, Gaukel, Eric, Hauser, Deirdre, Park, Seong Hee, Schock, Sara, Yardley, Vanessa, Randolph, Ryan, Plattner, Jacob J., Merchant, Tejal, Croft, Simon L., Jacobs, Robert T., Wring, S

Journal:

Antimicrobial Agents and Chemotherapy

Year:

2018

Language:

english

File:

PDF, 1.67 MB

english, 2018

2

Discovery and structure–activity study of a novel benzoxaborole anti-inflammatory agent (AN2728) for the potential topical treatment of psoriasis and atopic dermatitis

Tsutomu Akama, Stephen J. Baker, Yong-Kang Zhang, Vincent Hernandez, Huchen Zhou, Virginia Sanders, Yvonne Freund, Richard Kimura, Kirk R. Maples, Jacob J. Plattner

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 434 KB

english, 2009

3

Synthesis and structure–activity relationships of novel benzoxaboroles as a new class of antimalarial agents

Yong-Kang Zhang, Jacob J. Plattner, Yvonne R. Freund, Eric E. Easom, Yasheen Zhou, Jiri Gut, Philip J. Rosenthal, David Waterson, Francisco-Javier Gamo, Inigo Angulo-Barturen, Min Ge, Zhiya Li, Lingch

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 801 KB

english, 2011

4

Synthesis and antiviral activities of the major metabolites of the HIV protease inhibitor ABT-378 (Lopinavir)

Hing L Sham, David A Betebenner, Thomas Herrin, Gondi Kumar, Ayda Saldivar, Sudthida Vasavanonda, Akhter Molla, Dale J Kempf, Jacob J Plattner, Daniel W Norbeck

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 127 KB

english, 2001

5

Synthesis and SAR of novel benzoxaboroles as a new class of β-lactamase inhibitors

Yi Xia, Kathy Cao, Yasheen Zhou, M.R.K. Alley, Fernando Rock, Manisha Mohan, Maliwan Meewan, Stephen J. Baker, Sarah Lux, Charles Z. Ding, Guofeng Jia, Maureen Kully, Jacob J. Plattner

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 360 KB

english, 2011

6

Synthesis and structure–activity relationships of a novel series of HIV-1 protease inhibitors encompassing ABT-378 (Lopinavir)

Hing L. Sham, David A. Betebenner, Xiaoqi Chen, Ayda Saldivar, Sudthida Vasavanonda, Dale J. Kempf, Jacob J. Plattner, Daniel W. Norbeck

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 89 KB

english, 2002

7

Benzoxaboroles: a new class of potential drugs for human African trypanosomiasis

Jacobs, Robert T, Plattner, Jacob J, Nare, Bakela, Wring, Stephen A, Chen, Daitao, Freund, Yvonne, Gaukel, Eric G, Orr, Matthew D, Perales, Joe B, Jenks, Matthew

Journal:

Future Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 2.10 MB

english, 2011

8

Synthesis and SAR of acyclic HCV NS3 protease inhibitors with novel P4-benzoxaborole moieties

Xianfeng Li, Suoming Zhang, Yong-Kang Zhang, Yang Liu, Charles Z. Ding, Yasheen Zhou, Jacob J. Plattner, Stephen J. Baker, Wei Bu, Liang Liu, Wieslaw M. Kazmierski, Maosheng Duan, Richard M. Grimes, L

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 1.21 MB

english, 2011

9

Synthesis and biological evaluations of P4-benzoxaborole-substituted macrocyclic inhibitors of HCV NS3 protease

Charles Z. Ding, Yong-Kang Zhang, Xianfeng Li, Yang Liu, Suoming Zhang, Yasheen Zhou, Jacob J. Plattner, Stephen J. Baker, Liang Liu, Maosheng Duan, Richard L. Jarvest, Jingjing Ji, Wieslaw M. Kazmier

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 663 KB

english, 2010

10

An efficient synthesis for a new class antimalarial agent, 7-(2-carboxyethyl)-1,3-dihydro-1-hydroxy-2,1-benzoxaborole

Yong-Kang Zhang, Jacob J. Plattner, Eric E. Easom, David Waterson, Min Ge, Zhiya Li, Lingchao Li, Yong Jian

Journal:

Tetrahedron Letters

Year:

2011

Language:

english

File:

PDF, 313 KB

english, 2011

11

Benzoxaborole antimalarial agents. Part 2: Discovery of fluoro-substituted 7-(2-carboxyethyl)-1,3-dihydro-1-hydroxy-2,1-benzoxaboroles

Yong-Kang Zhang, Jacob J. Plattner, Yvonne R. Freund, Eric E. Easom, Yasheen Zhou, Long Ye, Huchen Zhou, David Waterson, Francisco-Javier Gamo, Laura M. Sanz, Min Ge, Zhiya Li, Lingchao Li, Hailong Wa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2012

Language:

english

File:

PDF, 848 KB

english, 2012

12

Identification of a 4-fluorobenzyl l -valinate amide benzoxaborole ( AN11736 ) as a potential development candidate for the treatment of Animal African Trypanosomiasis (AAT)

Akama, Tsutomu, Zhang, Yong-Kang, Freund, Yvonne R., Berry, Pamela, Lee, Joanne, Easom, Eric E., Jacobs, Robert T., Plattner, Jacob J., Witty, Michael J., Peter, Rosemary, Rowan, Tim G., Gillingwater,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2017

Language:

english

File:

PDF, 981 KB

english, 2017

13

Growing Organic Rabbiteye Blueberries in Georgia, USA: Results of Two Multi-Year Field Studies

Tertuliano, M., Krewer, G., Smith, J. E., Plattner, K., Clark, J., Jacobs, J., Andrews, E., Stanaland, D., Andersen, P., Liburd, O., Fonsah, E. G., Scherm, H.

Journal:

International Journal of Fruit Science

Year:

2012

Language:

english

File:

PDF, 153 KB

english, 2012

14

Crystal Structures of the Human and Fungal Cytosolic Leucyl-tRNA Synthetase Editing Domains: A Structural Basis for the Rational Design of Antifungal Benzoxaboroles

Elena Seiradake, Weimin Mao, Vincent Hernandez, Stephen J. Baker, Jacob J. Plattner, M.R.K. Alley, Stephen Cusack

Journal:

Journal of Molecular Biology

Year:

2009

Language:

english

File:

PDF, 1.86 MB

english, 2009

15

Synthesis of isotopically labelled [3-14C]- and [3,3-2H2]-5-fluoro-1,3-dihydro-1-hydroxy-2,1-benzoxaborole (AN2690), a new antifungal agent for the potential treatment of onychomycosis

Stephen J. Baker, Yong-Kang Zhang, Tsutomu Akama, Conrad Wheeler, Jacob J. Plattner, Richard M. Rosser, Ronald P. Reid, Neil S. Nixon

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2007

Language:

english

File:

PDF, 113 KB

english, 2007

16

Benzoxaborole Antimalarial Agents. Part 5. Lead Optimization of Novel Amide Pyrazinyloxy Benzoxaboroles and Identification of a Preclinical Candidate

Zhang, Yong-Kang, Plattner, Jacob J., Easom, Eric E., Jacobs, Robert T., Guo, Denghui, Freund, Yvonne R., Berry, Pamela, Ciaravino, Vic, Erve, John C. L., Rosenthal, Philip J., Campo, Brice, Gamo, Fra

Journal:

Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 1.23 MB

english, 2017

17

Synthesis of new acylsulfamoyl benzoxaboroles as potent inhibitors of HCV NS3 protease

Xianfeng Li, Yong-Kang Zhang, Yang Liu, Suoming Zhang, Charles Z. Ding, Yasheen Zhou, Jacob J. Plattner, Stephen J. Baker, Liang Liu, Wei Bu, Wieslaw M. Kazmierski, Lois L. Wright, Gary K. Smith, Rich

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 668 KB

english, 2010

18

Synthesis of novel benzoxaborole-containing phenylalanine analogues

Xianfeng Li, Jacob J. Plattner, Vincent Hernandez, Charles Z. Ding, Wei Wu, Yang Yang, Musheng Xu

Journal:

Tetrahedron Letters

Year:

2011

Language:

english

File:

PDF, 363 KB

english, 2011

19

Optimization of Isoxazoline Amide Benzoxaboroles for Identification of a Development Candidate as an Oral Long Acting Animal Ectoparasiticide

Zhang, Yong-Kang, Plattner, Jacob J., Easom, Eric E., Akama, Tsutomu, Zhou, Yasheen, Hunter White, W., Defauw, Jean M., Winkle, Joseph R., Balko, Terry W., Cao, Jianxin, Ge, Zhixin, Yang, Jianzhang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 761 KB

english, 2016

20

Discovery of a New Boron-Containing Antifungal Agent, 5-Fluoro-1,3-dihydro-1-hydroxy-2,1- benzoxaborole (AN2690), for the Potential Treatment of Onychomycosis

Baker, Stephen J., Zhang, Yong-Kang, Akama, Tsutomu, Lau, Agnes, Zhou, Huchen, Hernandez, Vincent, Mao, Weimin, Alley, M. R. K., Sanders, Virginia, Plattner, Jacob J.

Journal:

Journal of Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 66 KB

english, 2006

21

Benzoxaborole antimalarial agents. Part 3: design and syntheses of (carboxy-13C-3,3-2H2)-labeled and (3-14C)-labeled 7-(2-carboxyethyl)-1,3-dihydro-1-hydroxy-2,1-benzoxaboroles

Yong-Kang Zhang, Jacob J. Plattner, Eric E. Easom, Liang Liu, Daniel M. Retz, Min Ge, Hui-Hong Zhou

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2012

Language:

english

File:

PDF, 283 KB

english, 2012

22

Benzoxaborole Antimalarial Agents. Part 4. Discovery of Potent 6-(2-(Alkoxycarbonyl)pyrazinyl-5-oxy)-1,3-dihydro-1-hydroxy-2,1-benzoxaboroles

Zhang, Yong-Kang, Plattner, Jacob J., Easom, Eric E., Jacobs, Robert T., Guo, Denghui, Sanders, Virginia, Freund, Yvonne R., Campo, Brice, Rosenthal, Philip J., Bu, Wei, Gamo, Francisco-Javier, Sanz,

Journal:

Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 653 KB

english, 2015

23

Discovery of an orally bioavailable isoxazoline benzoxaborole (AN8030) as a long acting animal ectoparasiticide

Zhang, Yong-Kang, Plattner, Jacob J., Easom, Eric E., Zhou, Yasheen, Akama, Tsutomu, Bu, Wei, White, W. Hunter, Defauw, Jean M., Winkle, Joseph R., Balko, Terry W., Guo, Shenghai, Xue, Jian, Cao, Jian

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 624 KB

english, 2015

24

Peptide analogues of angiotensinogen effect of peptide chain length on renin inhibition

Jacob J. Plattner, Jonathan Greer, Anthony K.L. Fung, Herman Stein, Hollis D. Kleinert, Hing Leung Sham, Jill R. Smital, Thomas J. Perun

Journal:

Biochemical and Biophysical Research Communications

Year:

1986

Language:

english

File:

PDF, 474 KB

english, 1986

25

Synthesis of some DE and CDE ring analogs of camptothecin

Plattner, Jacob J., Gless, Richard D., Rapoport, Henry

Journal:

Journal of the American Chemical Society

Year:

1972

Language:

english

File:

PDF, 334 KB

english, 1972

26

Breast ductoscopy with a 0.55-mm microendoscope for direct visualization of intraductal lesions

VR Jacobs, M Kiechle, B Plattner, T Fischer, H Schaaf, S Paepke

Journal:

The Journal of the American Association of Gynecologic Laparoscopists

Year:

2004

Language:

english

File:

PDF, 119 KB

english, 2004

27

Novel Semisynthetic Derivative of Antibiotic Eremomycin Active against Drug-Resistant Gram-Positive Pathogens Including Bacillus anthracis †

Maples, Kirk R., Wheeler, Conrad, Ip, Emily, Plattner, Jacob J., Chu, Daniel, Zhang, Yong-Kang, Preobrazhenskaya, Maria N., Printsevskaya, Svetlana S., Solovieva, Svetlana E., Olsufyeva, Evgenia N., H

Journal:

Journal of Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 69 KB

english, 2007

28

Renin inhibitors. Design and synthesis of a new class of conformationally restricted analogs of angiotensinogen

Sham, Hing L., Bolis, Giorgio, Stein, Herman H., Fesik, Stephen W., Marcotte, Patrick A., Plattner, Jacob J., Rempel, Cheryl A., Greer, Jonathan

Journal:

Journal of Medicinal Chemistry

Year:

1988

Language:

english

File:

PDF, 1.69 MB

english, 1988

29

Synthesis and antibacterial activity of novel C12 ethyl ketolides

Matthew T. Burger, Christy Hiebert, Mehran Seid, Daniel T. Chu, Lynn Barker, Mike Langhorne, Ribhi Shawar, Jolene Kidney, Manoj C. Desai, Jacob J. Plattner

Journal:

Bioorganic & Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 287 KB

english, 2006

30

Novel macrocyclic HCV NS3 protease inhibitors derived from α-amino cyclic boronates

Xianfeng Li, Yong-Kang Zhang, Yang Liu, Charles Z. Ding, Yasheen Zhou, Qun Li, Jacob J. Plattner, Stephen J. Baker, Suoming Zhang, Wieslaw M. Kazmierski, Lois L. Wright, Gary K. Smith, Richard M. Grim

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 1.13 MB

english, 2010

31

Synthesis of dl-sirenin and dl-isosirenin

Bhalerao, Uday T., Plattner, Jacob J., Rapoport, Henry.

Journal:

Journal of the American Chemical Society

Year:

1970

Language:

english

File:

PDF, 731 KB

english, 1970

32

Nonpeptide renin inhibitors employing a novel 3-aza (or oxa)-2,4-dialkyl glutaric acid moiety as a P2/P3 amide bond replacement

Baker, William R., Fung, Anthony K. L., Kleinert, Hollis D., Stein, Herman H., Plattner, Jacob J., Armiger, Yoek Lin, Condon, Stephen L., Cohen, Jerome, Egan, David A.

Journal:

Journal of Medicinal Chemistry

Year:

1992

Language:

english

File:

PDF, 2.22 MB

english, 1992

33

[[(Aminomethyl)aryl]oxy]acetic acid esters. A new class of high-ceiling diuretics. 2. Modifications of the oxyacetic side chain

Plattner, Jacob J., Fung, Anthony K. L., Smital, Jill R., Lee, Cheuk Man, Crowley, Steven R., Pernet, Andre G., Bunnell, Paul R., Buckner, Steven A., Sennello, Lawrence T.

Journal:

Journal of Medicinal Chemistry

Year:

1984

Language:

english

File:

PDF, 1.32 MB

english, 1984

34

Synthesis of some DE and CDE ring analogs of camptothecin

Plattner, Jacob J., Gless, Richard D., Cooper, Geoffrey K., Rapoport, Henry

Journal:

Journal of Organic Chemistry

Year:

1974

Language:

english

File:

PDF, 1.39 MB

english, 1974

35

Chemical patents Profiting from Your Inventions

Mitscher, Lester A., Crowley, Steven R., Plattner, Jacob J.

Journal:

Analytical Chemistry

Year:

1994

Language:

english

File:

PDF, 9.61 MB

english, 1994

36

Synthesis and Antibacterial Activity of 6-Deoxysporeamicin A.

FAGHIH, RAMIN, FREIBERG, LESLIE, LEONARD, JAMES, PLATTNER, JACOB J., LARTEY, PAUL A.

Journal:

The Journal of Antibiotics

Year:

1996

Language:

english

File:

PDF, 162 KB

english, 1996

37

ChemInform Abstract: SYNTH. VON DL-SIRENIN UND DL-ISOSIRENIN

BHALERAO, UDAY T., PLATTNER, JACOB J., RAPOPORT, HENRY

Journal:

Chemischer Informationsdienst. Organische Chemie

Year:

1970

File:

PDF, 281 KB

1970

38

In Vitro penetration of a novel oxaborole antifungal (AN2690) into the human nail plate

Xiaoying Hui, Stephen J. Baker, Ronald C. Wester, Sherry Barbadillo, Anne K. Cashmore, Virginia Sanders, Karin M. Hold, Tsutomu Akama, Yong-Kang Zhang, Jacob J. Plattner, Howard I. Maibach

Journal:

Journal of Pharmaceutical Sciences

Year:

2007

Language:

english

File:

PDF, 195 KB

english, 2007

39

A practical stereoselective synthesis of (2S, 4S)-4-tert-butoxycarbonylamino-2-methylpyrrolidine

Qun Li, Daniel T.W. Chu, Kathleen Raye, Akiyo Claiborne, Louis Seif, Bryan Macri, Jacob J. Plattner

Journal:

Tetrahedron Letters

Year:

1995

Language:

english

File:

PDF, 314 KB

english, 1995

40

Renin inhibitors. Dipeptide analogs of angiotensinogen incorporating transition-state, nonpeptidic replacements at the scissile bond

Bolis, Giorgio, Fung, Anthony K. L., Greer, Jonathan, Kleinert, Hollis D., Marcotte, Patrick A., Perun, Thomas J., Plattner, Jacob J., Stein, Herman H.

Journal:

Journal of Medicinal Chemistry

Year:

1987

Language:

english

File:

PDF, 1.77 MB

english, 1987

41

Optimization and in vivo evaluations of a series of small, potent, and specific renin inhibitors containing a novel Leu-Val replacement

Dellaria, Joseph F., Maki, Robert G., Bopp, Barbara A., Cohen, Jerome, Kleinert, Hollis D., Luly, Jay R., Merits, Ilmar, Plattner, Jacob J., Stein, Herman H.

Journal:

Journal of Medicinal Chemistry

Year:

1987

Language:

english

File:

PDF, 1.08 MB

english, 1987

42

Preparation and in vitro and in vivo evaluation of quinolones with selective activity against Gram-positive organisms

Cooper, Curt S., Klock, Pamela L., Chu, Daniel T. W., Hardy, Dwight J., Swanson, Robert N., Plattner, Jacob J.

Journal:

Journal of Medicinal Chemistry

Year:

1992

Language:

english

File:

PDF, 984 KB

english, 1992

43

Synthesis and Activities of the Phosphonate Isostere of the Monophosphate of (±)Cyclobut-G

Norbeck, Daniel W., Sham, Hing L., Rosenbrook, William, Herrin, Thomas, Plattner, Jacob J.

Journal:

Nucleosides and Nucleotides

Year:

1992

Language:

english

File:

PDF, 363 KB

english, 1992

44

Highly potent and specific inhibitors of human renin

Hing L. Sham, Herman Stein, Cheryl A. Rempel, Jerome Cohen, Jacob J. Plattner

Journal:

Year:

1987

Language:

english

File:

PDF, 176 KB

english, 1987

45

Macrofilaricidal Benzimidazole-Benzoxaborole Hybrids as an Approach to the Treatment of River Blindness. Part 1. Amide Linked Analogs.

Akama, Tsutomu, Freund, Yvonne T., Berry, Pamela, Carter, David S., Easom, Eric E., Jarnagin, Kurt, Lunde, Christopher S., Plattner, Jacob J., Rock, Fernando, Stefanakis, Rianna, Fischer, Chelsea, Bul

Journal:

ACS Infectious Diseases

Year:

2019

File:

PDF, 304 KB

2019

46

Synthesis and evaluation of novel α-amino cyclic boronates as inhibitors of HCV NS3 protease

Xianfeng Li, Yong-Kang Zhang, Yang Liu, Charles Z. Ding, Qun Li, Yasheen Zhou, Jacob J. Plattner, Stephen J. Baker, Xuelei Qian, Dazhong Fan, Liang Liao, Zhi-Jie Ni, Gemma V. White, Jackie E. Mordaunt

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 1.37 MB

english, 2010

47

Novel lopinavir analogues incorporating non-Aromatic P-1 side chains—Synthesis and structure–Activity relationships

Hing L Sham, Chen Zhao, Leping Li, David A Betebenner, Ayda Saldivar, Sudthida Vasavanonda, Dale J Kempf, Jacob J Plattner, Daniel W Norbeck

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 98 KB

english, 2002

48

Neuroleptic activity in 5-aryltetrahydro-.gamma.-carbolines

Harbert, Charles A., Plattner, Jacob J., Welch, Willard M., Weissman, Albert, Koe, B. Kenneth

Journal:

Journal of Medicinal Chemistry

Year:

1980

Language:

english

File:

PDF, 1.03 MB

english, 1980

49

Antitumor Activity of 9(R)-Dihydrotaxane Analogs

Klein, Larry L., Li, Leping, Maring, Clarence J., Yeung, Clinton M., Thomas, Sheela A., Grampovnik, David J., Plattner, Jacob J.

Journal:

Journal of Medicinal Chemistry

Year:

1995

Language:

english

File:

PDF, 1.33 MB

english, 1995

50

Novel Lopinavir Analogues Incorporating Heterocyclic Replacements of Six-Member Cyclic Urea. Synthesis and Structure—Activity Relationships.

Hing L. Sham, David A. Betebenner, William Rosenbrook, Thomas Herrin, Ayda Saldivar, Sudthida Vasavanonda, Jacob J. Plattner, Daniel W. Norbeck

Journal:

Year:

2004

File:

PDF, 70 KB

2004

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